Cancer Subtype | Gene | Drug |
Breast Cancer | AKT1 | Capivasertib + Fulvestrant |
BRAF | Dabrafenib + Trametinib |
ERBB2 | Ado-Trastuzumab Emtansine |
Lapatinib + Capecitabine, Lapatinib + Letrozole |
Margetuximab + Chemotherapy |
Neratinib, Neratinib + Capecitabine |
Trastuzumab + Pertuzumab + Chemotherapy |
Trastuzumab + Tucatinib + Capecitabine |
Trastuzumab Deruxtecan |
Trastuzumab, Trastuzumab + Chemotherapy |
ESR1 | Elacestrant |
NTRK1 | Entrectinib |
Larotrectinib |
NTRK2 | Entrectinib |
Larotrectinib |
NTRK3 | Entrectinib |
Larotrectinib |
Microsatellite Instability-High (MSI-H) | Pembrolizumab |
Tumor Mutational Burden-High (TMB-H) | Pembrolizumab |
PIK3CA | Alpelisib + Fulvestrant |
Capivasertib + Fulvestrant |
PTEN | Capivasertib + Fulvestrant |
RET | Selpercatinib |